Dr.
Tadashi Inoue
Research fellow of the Japan Society for the Promotion of Science
Education
1992; BS Tokyo College of Pharmacy, Tokyo
1994; MS Tokyo College of Pharmacy, Tokyo
1997; Ph-D Tokyo University of Pharmacy and Life Science, Tokyo
Publication List
1) Catalytic Asymmetric Iodocarbocyclization Reaction of
4-Alkenylmalonates and Its Application to Enantiotopic Group
Selective Reaction, Inoue, Tadashi; Kitagawa,
Osamu; Saito, Akio; Taguchi, Takeo, J. Org. Chem. (1997),
62(21), 7384-7389
2) Fluoro-lactonization of 4-alkenoic acid derivatives with
N-fluoropentachloropyridinium triflate; Okada, Midori; Nakamura,
Yuko; Horikawa, Hiroaki; Inoue, Tadashi;
Taguchi, Takeo, J. Fluorine Chem. (1997),
82(2), 157-161
3) Iodocarbocyclization reaction; Kitagawa, Osamu; Inoue,
Tadashi; Taguchi, Takeo, Rev. Heteroat. Chem. (1996),
15, 243-262
4) Diastereoselective Iodocarbocyclization Reaction of 2- or
3-Oxy-4-pentenylmalonate Derivatives; Inoue, Tadashi;
Kitagawa, Osamu; Oda, Yoko; Taguchi, Takeo, J. Org. Chem.
(1996), 61(23), 8256-8263
5) Catalytic asymmetric iodocarbocyclization reaction; Inoue,
Tadashi; Kitagawa, Osamu; Ochiai, Orie; Shiro, Motoo;
Taguchi, Takeo, Tetrahedron Lett.
(1995), 36(51), 9333-6
6) Iodocarbocyclization reaction; Taguchi, Takeo; Kitagawa,
Osamu; Inoue, Tadashi. Yuki Gosei Kagaku
Kyokaishi (1995), 53(9), 770-9
7) Diastereoselective iodocarbocyclization reaction of
8-phenylmenthyl allylmalonate: an efficient preparation of a
synthetic intermediate of cyclopropaneamino acids; Inoue,
Tadashi; Kitagawa, Osamu; Ochiai, Orie; Taguchi, Takeo, Tetrahedron:
Asymmetry (1995), 6(3), 691-2
8) Enantioselective iodocarbocyclization of 4-alkenylmalonate
derivatives using a chiral titanium complex; Inoue,
Tadashi; Kitagawa, Osamu; Kurumizawa,
Shigeyuki; Ochiai, Orie; Taguchi, Takeo, Tetrahedron Lett.
(1995), 36(9), 1479-82
9) Diels-Alder reaction of N-allylic enamides and lactam
derivatives through iodine mediated activation; Kitagawa, Osamu;
Aoki, Katsuyuki; Inoue, Tadashi;
Taguchi, Takeo, Tetrahedron Lett. (1995),
36(4), 593-6
10) Diastereoselective iodocarbocyclization of 4-pentenylmalonate
derivatives: application to cyclosarkomycin synthesis, Kitagawa,
Osamu; Inoue, Tadashi;
Taguchi, Takeo, Tetrahedron Lett. (1994),
35(7), 1059-62
11) Ionic iodocarbocyclization reactions of 4-alkenyl- and
4-alkynylmalonate derivatives; Kitagawa, Osamu; Inoue,
Tadashi; Hirano, Keiko; Taguchi,
Takeo, J. Org. Chem. (1993), 58(11),
3106-12
12) Ionic iodocarbocyclization reaction; Kitagawa, Osamu; Inoue,
Tadashi; Taguchi, Takeo, Tetrahedron Lett. (1992),
33(16), 2167-70
13) A facile .a.-iodination reaction of unsaturated amides,
Kitagawa, Osamu; Hanano, Tokushi; Hirata, Tatsuya; Inoue,
Tadashi; Taguchi, Takeo,
Tetrahedron Lett. (1992), 33(10),
1299-302
Presentations
1. Lin, S.; Inoue, T.; Chakravarty, S.; Ojima, I. "Design and Synthesis of Taxoid-Epothilone Hybrids. Part I." 216th American Chemical Society National Meeting, August 23-27, 1998, Boston, Massachusetts; Abstr. ORGN 464.
2. Inoue, T.; Lin, S.; Walsh, J. J.; Borella, C.; Chakravarty, S.; Ojima, I. "Design and Synthesis of Taxoid-Epothilone Hybrids. Part II." 216th American Chemical Society National Meeting, August 23-27, 1998, Boston, Massachusetts; Abstr. ORGN380.
3. Lin, S.; Inoue, T.; Borella, C.; Walsh, J. J.; Chakravarty, S.; Ojima, I. "Design and Structure-Activity Relationship Study of Taxoid-Epothilone Hybrids." 216th American Chemical Society National Meeting, August 23-27, 1998, Boston, Massachusetts; Abstr. MEDI 313.